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US11098061, Compound III-1 PubChem CID 86301040
C=CC(=O)Nc1cc(-c2ccc3c(ccc4sc5c(c43)NC[C@@H](C)NC5=O)n2)cnc1C -
US11098061, Compound III-d-1 PubChem CID 86301505
C=CC(=O)Nc1cc(-c2cc(-c3cc4c(s3)C(=O)N[C@H](C)CN4)ccn2)ccc1OCCOC -
(R)—N-(3-acrylamido-4-(1-methylpiperidin-4-yl)phenyl)-3-methyl-5-oxo-2,3,4,5-tetrahydro-1H-benzo[4,5]thieno[3,2-e][1,4]diazepine-9-carboxamide PubChem CID 117610995
C=CC(=O)Nc1cc(NC(=O)c2ccc3sc4c(c3c2)NC[C@@H](C)NC4=O)ccc1C1CCN(C)CC1 -
N-[5-[(15R)-15-methyl-13-oxo-11-thia-6,14,17-triazatetracyclo[8.8.0.02,7.012,18]octadeca-1(10),2(7),3,5,8,12(18)-hexaen-5-yl]-2-(trifluoromethyl)phenyl]prop-2-enamide PubChem CID 117611197
C=CC(=O)Nc1cc(-c2ccc3c(ccc4sc5c(c43)NC[C@@H](C)NC5=O)n2)ccc1C(F)(F)F -
(3R)-3-methyl-5-oxo-N-[3-(prop-2-enoylamino)-4-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydro-[1]benzothiolo[3,2-e][1,4]diazepine-9-carboxamide PubChem CID 117611297
C=CC(=O)Nc1cc(NC(=O)c2ccc3sc4c(c3c2)NC[C@@H](C)NC4=O)ccc1C(F)(F)F -
N-[5-[(15R)-15-methyl-13-oxo-11-thia-6,14,17-triazatetracyclo[8.8.0.02,7.012,18]octadeca-1(10),2(7),3,5,8,12(18)-hexaen-5-yl]-2-(trifluoromethoxy)phenyl]prop-2-enamide PubChem CID 117611303
C=CC(=O)Nc1cc(-c2ccc3c(ccc4sc5c(c43)NC[C@@H](C)NC5=O)n2)ccc1OC(F)(F)F -
(R)—N-(5-(10-methyl-8-oxo-9,10,11,12-tetrahydro-8H-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-3-yl)-2-(1-methylpiperidin-4-yl)phenyl)acrylamide PubChem CID 117611317
C=CC(=O)Nc1cc(-c2ccc3c(ccc4sc5c(c43)NC[C@@H](C)NC5=O)n2)ccc1C1CCN(C)CC1