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US10774071, Example B-31 PubChem CID 146297332
COc1nc(-c2cccc(-c3cccc4c3CC[C@@H]4Oc3nc(OCc4cc(Cl)cc(C#N)c4)c(CN4CC5(C(=O)O)CCC4CC5)cc3Cl)c2Cl)ccc1CNC[C@@H]1CCC(=O)N1