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US10125148, Example 6 PubChem CID 118334301
CCc1ccc2c(c1)-c1cccc(c1)-c1cc3nc(C)c([C@H](OC(C)(C)C)C(=O)O)c(n3n1)N1CCC(C)(CC1)OC/C=C/C[C@H](C)O2