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(S)-N-(1-(3-chloro-4-fluorophenyl)-2,2,2-trifluoroethyl)-5-cyano-N-ethylpyridine-3-sulfonamide (Example PubChem CID 168898591
CCN(C(c1ccc(F)c(Cl)c1)C(F)(F)F)S(=O)(=O)c1cncc(C#N)c1 -
(R)-N-ethyl-N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)pyrimidine-5-sulfonamide (Example 133) and (R) PubChem CID 168898599
CCN(C(c1ccc(F)cc1)C(F)(F)F)S(=O)(=O)c1cncnc1 -
(S)-N-ethyl-2-methyl-N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)pyrimidine-5-sulfonamide (Example 76) PubChem CID 168898698
CCN(C(c1ccc(F)cc1)C(F)(F)F)S(=O)(=O)c1cnc(C)nc1 -
(S)-5-cyano-N-ethyl-N-(2,2,2-trifluoro-1-(4-fluoro-3-methoxyphenyl)ethyl)pyridine-3-sulfonamide (Example PubChem CID 168898755
CCN(C(c1ccc(F)c(OC)c1)C(F)(F)F)S(=O)(=O)c1cncc(C#N)c1 -
N-ethyl-N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)imidazo[1,2-a]pyridine-7-sulfonamide (Example 135) PubChem CID 168898868
CCN(C(c1ccc(F)cc1)C(F)(F)F)S(=O)(=O)c1ccn2ccnc2c1 -
(S)-N,5-dimethyl-N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)thiophene-2-sulfonamide (Example 12) and PubChem CID 168899084
Cc1ccc(S(=O)(=O)N(C)[C@H](c2ccc(F)cc2)C(F)(F)F)s1 -
N,N-dimethyl-5-(N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)sulfamoyl)thiophene-2-carboxamide (Example PubChem CID 168899202
CN(C)C(=O)c1ccc(S(=O)(=O)NC(c2ccc(F)cc2)C(F)(F)F)s1 -
(S)-5-cyano-N-ethyl-N-(2,2,2-trifluoro-1-(4-fluoro-3-methylphenyl)ethyl)pyridine-3-sulfonamide (Example PubChem CID 169784685
CCN(C(c1ccc(F)c(C)c1)C(F)(F)F)S(=O)(=O)c1cncc(C#N)c1 -
(R)-3-chloro-N-methyl-N-(2,2,2-trifluoro-1-(4-(trifluoromethyl)phenyl)ethyl)imidazo[1,2-a]pyridine-6- PubChem CID 169795021
CN(C(c1ccc(C(F)(F)F)cc1)C(F)(F)F)S(=O)(=O)c1ccc2ncc(Cl)n2c1 -
(R)-5-cyano-N-methyl-N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)thiophene-2-sulfonamide (Example 6) and PubChem CID 169931800
CN([C@H](c1ccc(F)cc1)C(F)(F)F)S(=O)(=O)c1ccc(C#N)s1 -
(R)-5-cyano-N-methyl-N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)thiophene-2-sulfonamide (Example 6) and PubChem CID 169933333
CN([C@@H](c1ccc(F)cc1)C(F)(F)F)S(=O)(=O)c1ccc(C#N)s1 -
2-methyl-4-(((R)-1-(2-methyl-3-(trifluoromethyl)phenyl)ethyl)amino)-6-((S)-3-methyltetrahydrofuran-3- PubChem CID 169972468
C[C@@H](Nc1nn(C)c(=O)c2cc(=O)n([C@]3(C)CCOC3)cc12)c1cccc(C(F)(F)F)c1F -
(R)-6-(1-((6-cyclopropyl-2-methyl-1,7-dioxo-1,2,6,7-tetrahydropyrido[3,4-d]pyridazin-4-yl)amino)ethyl PubChem CID 170776070
Cc1cc([C@H](C)Nc2nn(C)c(=O)c3cc(=O)n(C4CC4)cc23)cc2c1c(C#N)nn2C -
6-cyclopropyl-2-methyl-4-(((R)-1-(2-methyl-3-(trifluoromethyl)phenyl)ethyl)amino)-8-((S)-pyrrolidin-2 PubChem CID 170776075
Cc1c([C@@H](C)Nc2nn(C)c(=O)c3c([C@H]4CCCN4)c(=O)n(C4CC4)cc23)cccc1C(F)(F)F -
6-[(1S,2R)-2-(5-fluoro-3-pyridyl)cyclopropyl]-2-methyl-4-[[(1R)-1-[2-methyl-3-(trifluoromethyl)phenyl PubChem CID 170776080
Cc1c([C@@H](C)Nc2nn(C)c(=O)c3cc(=O)n([C@@H]4C[C@H]4c4cncc(F)c4)cc23)cccc1C(F)(F)F -
4-(((R)-1-(3-(difluoromethyl)-2-fluorophenyl)ethyl)amino)-2-methyl-6-((R)-3-(trifluoromethyl)pyrrolidin PubChem CID 172122141
C[C@@H](CNc1nn(C)c(=O)c2cc(=O)n([C@@]3(C(F)(F)F)CCNC3)cc12)c1cccc(C(F)F)c1F -
(R)-N-methyl-N-(2,2,2-trifluoro-1-(4-(trifluoromethyl)phenyl)ethyl)-[1,2,4]triazolo[1,5-a]pyridine-7- PubChem CID 172216088
CN([C@H](c1ccc(C(F)(F)F)cc1)C(F)(F)F)S(=O)(=O)c1ccn2ncnc2c1 -
(R)-N-ethyl-N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazine PubChem CID 175901534
CCN(C(c1ccc(F)cc1)C(F)(F)F)S(=O)(=O)c1ccc2nnc(C)n2n1 -
(R)-N-ethyl-2,2-difluoro-N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)benzo[d][1,3]dioxole-5-sulfonamide PubChem CID 175901572
CCN(C(c1ccc(F)cc1)C(F)(F)F)S(=O)(=O)c1ccc2c(c1)OC(F)(F)O2 -
5-fluoro-N-methyl-N-(2,2,2-trifluoro-1-(4-fluorophenyl)ethyl)thiophene-2-sulfonamide (Example 18) and PubChem CID 176509317
C[C@H](c1ccc(F)cc1)N(C)S(=O)(=O)c1ccc(F)s1