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(R)-N-(1-Acryloylpiperidin-3-yl)-5-(2'',3''-difluoro-[1,1''-biphenyl]-3- yl)-4-oxo-4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2- carboxamide; PubChem CID 155922869
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(-c5cccc(F)c5F)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-5-(3''-fluoro-[1,1''-biphenyl]-3-yl)-4- oxo-4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2- carboxamide; PubChem CID 155922870
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(-c5cccc(F)c5)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-5-(2''-methyl-[1,1''-biphenyl]-3-yl)- 4-oxo-4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2- carboxamide; PubChem CID 155922871
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(-c5ccccc5C)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-4-oxo-5-(6-phenoxypyridin-3-yl)- 4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922872
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4ccc(Oc5ccccc5)nc4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-5-(3''-chloro-[1,1''-biphenyl]-3-yl)- 4-oxo-4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2- carboxamide; PubChem CID 155922873
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(-c5cccc(Cl)c5)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-5-(2''-chloro-[1,1''-biphenyl]-3-yl)- 4-oxo-4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2- carboxamide; PubChem CID 155922875
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(-c5ccccc5Cl)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-4-oxo-5-(5-phenoxypyridin-2-yl)- 4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922877
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4ccc(Oc5ccccc5)cn4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-5-(3-benzylphenyl)-4-oxo-4,5- dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922879
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(Cc5ccccc5)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-5-(3''-methyl-[1,1''-biphenyl]-3-yl)- 4-oxo-4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2- carboxamide; PubChem CID 155922880
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(-c5cccc(C)c5)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-5-(3-cyclohexylphenyl)-4-oxo-4,5- dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922881
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(C5CCCCC5)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-5-(2,2-difluorobenzo[d][1,3]dioxol- 5-yl)-4-oxo-4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2- carboxamide; PubChem CID 155922884
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4ccc5c(c4)OC(F)(F)O5)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-4-oxo-5-(3-phenoxyphenyl)-4,5- dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922886
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(Oc5ccccc5)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-4-oxo-5-(5-phenoxypyrazin-2-yl)- 4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922887
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cnc(Oc5ccccc5)cn4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-5-(3-isopropylphenyl)-4-oxo-4,5- dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922888
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(C(C)C)c4)C4CCNC(S2)C34)C1 -
(R)-5-([1,1''-Biphenyl]-3-yl)-N-(1-acryloylpyrrolidin-3-yl)-4-oxo-4,5- dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922889
C=CC(=O)N1CC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(-c5ccccc5)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-4-oxo-5-(3-propylphenyl)-4,5- dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922890
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(CCC)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-5-(3-cyclobutylphenyl)-4-oxo-4,5- dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922891
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(C5CCC5)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-4-oxo-5-(5-phenylpyridin-3-yl)- 4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922893
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cncc(-c5ccccc5)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-4-oxo-5-(3-(pyridin-3-yl)phenyl)- 4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922894
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(-c5cccnc5)c4)C4CCNC(S2)C34)C1 -
(R)-N-(1-Acryloylpiperidin-3-yl)-4-oxo-5-(3-(pyridin-2-yl)phenyl)- 4,5-dihydro-3H-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide; PubChem CID 155922896
C=CC(=O)N1CCC[C@@H](NC(=O)C2=C3NC(=O)N(c4cccc(-c5ccccn5)c4)C4CCNC(S2)C34)C1